| 1-{4-[3-(4-Fluorophenyl)-4,5-dihydroisoxazol-5-yl]butyl}-4-(2-methoxyphenyl)piperazine | C₂₄H₃₀FN₃O₂ | 411.521 g/mol |
| 1-{4-[3-(8-Amino-1-iodoimidazo[1,5-a]pyrazin-3-yl)cyclobutyl]piperazin-1-yl}ethanone | C₁₆H₂₁IN₆O | 440.289 g/mol |
| 1-{4-[3-(8-Chloro-1-iodoimidazo[1,5-a]pyrazin-3-yl)cyclobutyl]piperazin-1-yl}ethanone | C₁₆H₁₉ClIN₅O | 459.719 g/mol |
| 1-{4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}-2-propanone | C₁₇H₁₇F₃N₂O | 322.33 g/mol |
| 1-{4-[4-(1-Ethyl-propylamino)-3,6-dimethyl-pyridin-2-yloxy]-3,5-dimethyl-phenyl}-ethanol | C₂₂H₃₂N₂O₂ | 356.51 g/mol |
| 1-{4-[4-(2-Chloro-5-nitro-benzoyl)-piperazin-1-yl]-3-fluoro-phenyl}-ethanone | C₁₉H₁₇ClFN₃O₄ | 405.813 g/mol |
| 1-{4-[4-(2-Phenylethyl)-1,3-thiazol-2-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethanone | C₂₂H₂₄N₂OS₂ | 396.581 g/mol |
| 1-{4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl}-1H-benzimidazole | C₁₉H₂₄N₆ | 336.443 g/mol |
| 1-{4-[4-(3-chloropropoxy)phenyl]tetrahydro-2H-pyran-4-yl}-N,N-dimethylmethanamine | C₁₇H₂₆ClNO₂ | 311.853 g/mol |
| 1-{4-[4-(3-Pyrrolidin-1-ylpropoxy)phenyl]tetrahydropyran-4-ylmethyl)pyrrolidin-3-ol | C₂₃H₃₆N₂O₃ | 388.552 g/mol |
| 1-{4-[4-(3-thiomorpholin-4-ylpropoxy)phenyl]tetrahydro-2H-pyran-4-yl}methanamine | C₁₉H₃₀N₂O₂S | 350.528 g/mol |
| 1-{4-[4-(4-Methanesulfonyl-phenoxy)-pyrazolo[3,4-d]pyrimidin-1-yl]-piperidin-1-yl}-2,2-dimethyl-propan-1-one | C₂₂H₂₇N₅O₄S | 457.556 g/mol |
| 1-{4-[4-(4-Methanesulfonyl-phenoxy)-pyrazolo[3,4-d]pyrimidin-1-yl]-piperidin-1-yl}-3,3-dimethyl-butan-1-one | C₂₃H₂₉N₅O₄S | 471.583 g/mol |
| 1-{4-[4-(Azetidin-3-ylamino)-6-morpholin-4-yl-1,3,5-triazin-2-yl]phenyl}-3-(4-methylphenyl)urea | C₂₄H₂₈N₈O₂ | 460.542 g/mol |
| 1-{4-[4-(Tert-butoxycarbonyl)piperazin-1-yl]-2-fluorophenyl}cyclopropanecarboxylic acid | C₁₉H₂₅FN₂O₄ | 364.417 g/mol |
| 1-{4-[4-Amino-7-(2-bromoethyl)pyrrolo[2,1-f][1,2,4]triazin-5-yl]-2-fluorophenyl}-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | C₂₂H₁₆BrF₅N₆O | 555.305 g/mol |
| 1-{4-[4-Amino-7-(4-hydroxybutyl)pyrrolo[2,1-f][1,2,4]triazin-5-yl]-2-fluorophenyl}-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | C₂₄H₂₁F₅N₆O₂ | 520.462 g/mol |
| 1-{4-[4-Amino-7-(4-{[tert-butyl(dimethyl)silyl]oxy}butyl)pyrrolo[2,1-f][1,2,4]triazin-5-yl]-2-fluorophenyl}-3-[2-fluoro-5-(trifluoromethyl)-phenyl]urea | C₃₀H₃₅F₅N₆O₂Si | 634.726 g/mol |
| 1-{4-[4-Hydroxy-2-(4-methylphenyl)benzoylamino]benzoyl}-1,2,3,4-tetrahydroquinoline | C₃₀H₂₆N₂O₃ | 462.549 g/mol |
| 1-{4-[4-Methoxy-2-(4-methylphenyl)benzoylamino]benzoyl}-1,2,3,4-tetrahydroquinoline | C₃₁H₂₈N₂O₃ | 476.576 g/mol |
| 1-{4-[4-morpholin-4-yl-6-(tetrahydro-2H-pyran-4-yloxy)-1,3,5-triazin-2-yl]phenyl}-3-phenylurea | C₂₅H₂₈N₆O₄ | 476.537 g/mol |
| 1-{4-[5-(3,4-Dichlorobenzoylamino)pyridin-2-yloxy]benzoyl}piperidine-4-carboxylic acid | C₂₅H₂₁Cl₂N₃O₅ | 514.365 g/mol |
| 1-{4-[5-(3,5-dichloro-phenyl)-5-trifluoromethyl-4,5-dihydro-isoxazol-3-yl]-naphthalen-1-yl}-1H-[1,2,4]triazole | C₂₂H₁₃Cl₂F₃N₄O | 477.273 g/mol |
| 1-{4-[5-(4-Isopropyl-piperazine-1-carbonyl)-1H-indole-2-carbonyl]-piperazin-1-yl}-2-methyl-propan-1-one | C₂₅H₃₅N₅O₃ | 453.587 g/mol |
| 1-{4-[5-(4-{2-[Bis-(4-methoxy-benzyl)-amino]-pyrimidin-5-yl}-2-morpholin-4-yl-5,6-dihydro-pyrrolo[2,3-d]pyrimidin-7-yl)-pyridin-2-yl]-piperazin-1-yl}-ethanone | C₄₁H₄₆N₁₀O₄ | 742.885 g/mol |
| 1-{4-[6-(1-Methylethyl)-5,6,7,8-tetrahydropyrazolo[3,4-d]azepin-2(4H)-yl]phenyl}-2-pyrrolidinone | C₂₀H₂₆N₄O | 338.455 g/mol |
| 1-{4-[6-(2-Hydroxy-ethylamino)-pyrimidin-4-yloxy]-phenyl}-3-(3-trifluoromethyl-phenyl)-urea | C₂₀H₁₈F₃N₅O₃ | 433.39 g/mol |
| 1-{4-[6-(4-Methanesulfonyl-phenylamino)-5-nitro-pyrimidin-4-yloxy]-piperidin-1-yl}-3,3-dimethyl-butan-2-one | C₂₂H₂₉N₅O₆S | 491.57 g/mol |
| 1-{4-[6-Fluoro-2-phenoxymethyl-3-(4-trifluoromethoxy-benzyl)-3H-benzoimidazol-5-yl]-piperazin-1-yl}-butan-1-one | C₃₀H₃₀F₄N₄O₃ | 570.587 g/mol |
| 1-{4-[7-(1-Acetylpyrrolidin-3-yl)-4-aminopyrrolo[2,1-f][1,2,4]triazin-5-yl]phenyl}-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | C₂₆H₂₃F₄N₇O₂ | 541.509 g/mol |
| 1-{4-[7-(2-Chloroethoxy)-6-methoxy-quinolin-4-yloxy]-2-fluorophenyl}-3-(3,3-dimethyl-butyl)urea | C₂₅H₂₉ClFN₃O₄ | 489.975 g/mol |
| 1-{4-[7-(4-Methanesulfonyl-phenyl)-imidazo[1,2-a]pyridin-3-yl]-benzyl}-3-(3-trifluoromethyl-phenyl)-urea | C₂₉H₂₃F₃N₄O₃S | 564.589 g/mol |
| 1-{4-[N-(pyridin-3-ylmethoxycarbonyl)aminomethyl]benzoyl}imidazole | C₁₈H₁₆N₄O₃ | 336.351 g/mol |
| 1-{4-Aminopyrrolo[2,1-f][1,2,4]triazin-7-yl}-2-chloroethan-1-one | C₈H₇ClN₄O | 210.624 g/mol |
| 1-{4-Chloro-2-[(4-chloro-2-methoxy-6-methylphenyl)amino]-1-methyl-1H-benzimidazol-7-yl}-2,2-dimethylpropan-1-one | C₂₁H₂₃Cl₂N₃O₂ | 420.34 g/mol |
| 1-{4-Methoxy-3-[2-(3-oxetan-3-yl-phenyl)-ethoxy]-benzoylamino}-4-trifluoromethyl-cyclohexanecarboxylic Acid | C₂₇H₃₀F₃NO₆ | 521.532 g/mol |
| 1-{4-Methoxy-3-[2-(3-oxetan-3-yl-phenyl)-ethoxy]-benzoylamino}-4-trifluoromethyl-cyclohexanecarboxylic Acid Methyl Ester | C₂₈H₃₂F₃NO₆ | 535.559 g/mol |
| 1-{4-methyl-5-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}ethanol | C₁₂H₁₂F₃N₃O | 271.242 g/mol |
| 1-{4-Nitro-3-[(2,2,2-trifluoroethyl)oxy]phenyl}-4-piperidinol | C₁₃H₁₅F₃N₂O₄ | 320.267 g/mol |
| 1-{4-Nitro-3-[(2,2,2-trifluoroethyl)oxy]phenyl}-4-piperidinone | C₁₃H₁₃F₃N₂O₄ | 318.251 g/mol |
| 1-{4-{2-[N-(trans-4-methylcyclohexyl) carbamoyl]ethyl}-2-methoxyphenoxyacetyl}-4-piperidinopiperidine | C₂₉H₄₅N₃O₄ | 499.696 g/mol |
| 1-{4-{2-[N-(trans-4-methylcyclohexyl)carbamoyl]vinyl}-2-methoxyphenoxyacetyl}-4-piperidinopiperidine | C₂₉H₄₃N₃O₄ | 497.68 g/mol |
| 1-{5'-[3,4-Bis(benzoyloxymethyl)benzyloxy]-2'methyl-2-propylbiphenyl-4-yl}-1-propanone | C₄₂H₄₀O₆ | 640.776 g/mol |
| 1-{5'-[3,4-Bis(benzoyloxymethyl)benzyloxy]-2,2'-diethylbiphenyl-4-yl}-1-propanone | C₄₂H₄₀O₆ | 640.776 g/mol |
| 1-{5-(Tert-butyl)-2-[(6,7-dimethoxy-4-quinolyl)oxy]phenyl}-1-propanol | C₂₄H₂₉NO₄ | 395.499 g/mol |
| 1-{5-(Tert-butyl)-2-[(6,7-dimethoxy-4-quinolyl)oxy]phenyl}-1-propanone | C₂₄H₂₇NO₄ | 393.483 g/mol |
| 1-{5-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridin-2-yl}-1H-pyrrolo[2,3-c]pyridine | C₁₈H₁₂N₄S | 316.389 g/mol |
| 1-{5-[1-(1,3-Dimethoxypropan-2-yl)-4-oxo-3-(piperazin-1-ylcarbonyl)-1,4-dihydroquinolin-6-yl]-4-[4-(trifluoromethyl)-1,3-thiazol-2-yl]pyridin-2-yl}-3-ethylurea | C₃₁H₃₄F₃N₇O₅S | 673.718 g/mol |
| 1-{5-[1-(4-Chloro-2-trifluoromethyl-benzyl)-1H-indazol-5-ylmethylene]-4-oxo-4,5-dihydro-thiazol-2-yl}piperidine-4-carboxylic acid | C₂₅H₂₀ClF₃N₄O₃S | 548.974 g/mol |
| 1-{5-[1-(4-Methoxy-2-trifluoromethyl-benzyl)-1H-indazol-5-ylmethylene]-4-oxo-4,5-dihydro-thiazol-2-yl}-azetidine-3-carboxylic acid | C₂₄H₁₉F₃N₄O₄S | 516.501 g/mol |
| 1-{5-[2-(Thieno[3,2-d]pyrimidin-4-yloxy)-1-triisopropylsilanyloxymethyl-ethyl]-thiazol-2-yl}-3-(3-trifluoromethyl-phenyl)-urea | C₂₉H₃₆F₃N₅O₃S₂Si | 651.853 g/mol |
| 1-{5-[4-(2,2-Difluoro-cyclopropylmethyl)-piperazin-1-yl]-pyridin-2-yl}-1,2,3,4-tetrahydroquinoxaline | C₂₁H₂₅F₂N₅ | 385.462 g/mol |
| 1-{5-[5-(4-Chloro-phenyl)-pyridin-2-ylethynyl]-pyridin-2-yl}-4-methyl-piperazine | C₂₃H₂₁ClN₄ | 388.902 g/mol |
| 1-{5-[8-(1-Ethyl-propyl)-2,6-dimethyl-imidazo[1,2-b]pyridazin-3-yl]-4-methyl-thiazol-2-yl}-piperidin-4-one | C₂₂H₂₉N₅OS | 411.575 g/mol |
| 1-{5-Chloro-2-[(phenylmethyl)oxy]phenyl}ethanone | C₁₅H₁₃ClO₂ | 260.72 g/mol |
| 1-{5-Chloro-2-[4-(3,5-dimethylpyridin-2-yl)piperazine-1-carbonyl]phenyl}pyrrolidin-2-one | C₂₂H₂₅ClN₄O₂ | 412.921 g/mol |
| 1-{5-tert-Butyl-2-[2-(tert-butyl-dimethyl-silanyloxy)-ethyl]-2H-pyrazol-3-yl}-3-{4-[7-(4-methanesulfonyl-phenyl)-imidazo[1,2-a]pyridin-3-yl]-benzyl}-urea | C₃₇H₄₈N₆O₄SSi | 700.982 g/mol |
| 1-{6-[(1E)-N-(2,4,6-Trimethylphenyl)ethanimidoyl]pyridin-2-yl}ethan-1-one | C₁₈H₂₀N₂O | 280.371 g/mol |
| 1-{6-[(Diphenylmethylene)amino]naphthalen-2-yl}-2-methyl-1-(1-trityl-1H-imidazol-4-yl)-1-propanol | C₄₉H₄₁N₃O | 687.887 g/mol |
| 1-{6-[(Tert-butyldimethylsilanyl)ethynyl]pyridin-3-yl}-4-methylcyclohexanol | C₂₀H₃₁NOSi | 329.56 g/mol |
| 1-{6-[({[(1-methyl-1H-tetrazol-5-yl)(phenyl)methylene]amino}oxy)methyl]pyridin-2-yl}methanamine | C₁₆H₁₇N₇O | 323.36 g/mol |
| 1-{6-[1-(2-Chloro-4,6-dimethylphenylimino)ethyl]pyridin-2-yl}ethanone | C₁₇H₁₇ClN₂O | 300.789 g/mol |
| 1-{6-[2-Aminoethyl]pyridin-2-yl}-3-(2-pyridin-4-yl-thiazol-4-yl)urea | C₁₆H₁₆N₆OS | 340.412 g/mol |
| 1-{6-[2-Fluoro-4-(3-phenylacetylthioureido)phenoxy]pyrimidin-4-yl}-3-(1-methylpiperidin-4-yl)urea | C₂₆H₂₈FN₇O₃S | 537.621 g/mol |
| 1-{6-[4-(2-Trifluoromethylbenzoyl)piperazin-1-yl]pyridazin-3-yl}imidazolidin-2-one | C₁₉H₁₉F₃N₆O₂ | 420.395 g/mol |
| 1-{6-[4-(Trifluoromethyl)phenyl]-2-pyridinyl}-1-pentanol | C₁₇H₁₈F₃NO | 309.331 g/mol |
| 1-{6-Benzyloxy-1-[4-(2-pyrrolidin-1-yl-ethoxy)phenyl]-3,4-dihydro-1H-isoquinolin-2-yl}-2,2,2-trifluoroethanone | C₃₀H₃₁F₃N₂O₃ | 524.583 g/mol |
| 1-{[(2-Bromoethyl)oxy]methyl}-3-fluorobenzene | C₉H₁₀BrFO | 233.08 g/mol |
| 1-{[(2-Bromoethyl)oxy]methyl}-4-(1,1-dimethylethyl)benzene | C₁₃H₁₉BrO | 271.198 g/mol |
| 1-{[(2-Chloro-5,6-dimethyl-3-nitropyridin-4-yl)amino]methyl}cyclohexanol | C₁₄H₂₀ClN₃O₃ | 313.785 g/mol |
| 1-{[(2-Methylphenylcarbonyloxy)ethoxy]carbonylamino}cyclopropanecarboxylic Acid | C₁₅H₁₇NO₆ | 307.302 g/mol |
| 1-{[(2Z)-5-tert-butyl-2-{[(5-chloro-2-methoxyphenyl)(cyanoimino)methyl]imino}-1,3-thiazol-3(2H)-yl]methyl}cyclopentyl acetate | C₂₄H₂₉ClN₄O₃S | 489.041 g/mol |
| 1-{[(3-Amino[1,5]naphthyridin-4-yl)amino]methyl}cyclohexanol | C₁₅H₂₀N₄O | 272.352 g/mol |
| 1-{[(3-Nitro[1,5]naphthyridin-4-yl)amino]methyl}cyclohexanol | C₁₅H₁₈N₄O₃ | 302.334 g/mol |
| 1-{[(3-Nitroquinolin-4-yl)amino]methyl}cyclopentanol | C₁₅H₁₇N₃O₃ | 287.319 g/mol |
| 1-{[(6-Bromopyridin-2-yl)methyl]sulfonyl}-2-methylpropan-2-ol | C₁₀H₁₄BrNO₃S | 308.197 g/mol |
| 1-{[(9H-Fluoren-9-YL)methoxy]carbonyl}-4-hydroxypyrrolidine-2-carboxylic acid | C₂₀H₁₉NO₅ | 353.374 g/mol |
| 1-{[(Benzyloxy)(formyl)amino]methyl}cyclopentane-1-carboxylic acid | C₁₅H₁₉NO₄ | 277.32 g/mol |
| 1-{[(Benzyloxy)amino]methyl}-3-butylcyclobutane-1-carboxylic acid | C₁₇H₂₅NO₃ | 291.391 g/mol |
| 1-{[(Benzyloxy)amino]methyl}cycloheptane-1-carboxylic acid | C₁₆H₂₃NO₃ | 277.364 g/mol |
| 1-{[(Benzyloxy)amino]methyl}cyclopentane-1-carboxylic acid | C₁₄H₁₉NO₃ | 249.31 g/mol |
| 1-{[(Benzyloxy)imino]methyl}-3-butylcyclobutane-1-carboxylic acid | C₁₇H₂₃NO₃ | 289.375 g/mol |
| 1-{[(Benzyloxy)imino]methyl}cycloheptane-1-carboxylic acid | C₁₆H₂₁NO₃ | 275.348 g/mol |
| 1-{[(Tert-butyldimethylsilyl)oxy]methyl}cyclobutane-1-carbaldehyde | C₁₂H₂₄O₂Si | 228.408 g/mol |
| 1-{[(trans-4-{6-[(2'-cyanobiphenyl-4-yl)methyl]-5-oxo-7-propyl[1,2,4]triazolo[1,5-a]pyrimidin-4(5H)-yl}cyclohexyl)oxy]methyl}cyclobutanecarboxylic acid | C₃₄H₃₇N₅O₄ | 579.701 g/mol |
| 1-{[1,1'-Biphenyl]-4-yl}-2-bromoethan-1-ol | C₁₄H₁₃BrO | 277.161 g/mol |
| 1-{[1-(2-tert-Butoxycarbonylamino-3,3-dimethyl-butyryl)-4-(3-ethoxy-isoquinolin-1-yloxy)-pyrrolidine-2-carbonyl]-amino}-2-ethyl-cyclopropanecarboxylic acid | C₃₃H₄₆N₄O₈ | 626.751 g/mol |
| 1-{[1-(2-tert-Butoxycarbonylamino-3,3-dimethylbutyryl)-4-hydroxypyrrolidine-2-carbonyl]-amino}-2-ethyl-cyclopropanecarboxylic acid | C₂₂H₃₇N₃O₇ | 455.552 g/mol |
| 1-{[1-(3-Chlorophenyl)-5-(3-trifluoromethoxyphenyl)-1H-pyrazol-3-yl]carbonyl}piperazine | C₂₁H₁₈ClF₃N₄O₂ | 450.848 g/mol |
| 1-{[1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-1H-imidazol-4-yl]methyl}-4-(4-methylphenyl)-piperazine | C₂₇H₂₅Cl₃N₄ | 511.884 g/mol |
| 1-{[1-(4-Chlorophenyl)cyclopropyl]carbonyl}-3-(1,1-dimethylpropyl)pyrrolidin-3-ol | C₁₉H₂₆ClNO₂ | 335.875 g/mol |
| 1-{[1-(4-Iodophenyl)cyclopropyl]carbonyl}pyrrolidine | C₁₄H₁₆INO | 341.192 g/mol |
| 1-{[1-(6-Tri-fluoromethyl-pyridin-3-ylmethoxy)-naphthalene-2-carbonyl]-amino}-cyclobutane-carboxylic acid ethyl ester | C₂₅H₂₃F₃N₂O₄ | 472.463 g/mol |
| 1-{[1-(p-Chlorophenyl)cyclopropyl]methyl}-3-(2,6-dichlorobenzylideneamino)guanidine | C₁₈H₁₇Cl₃N₄ | 395.721 g/mol |
| 1-{[2-(1,1-difluoroethyl)-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]sulfonyl}-1H-pyrrole-3-carbaldehyde | C₂₀H₂₁F₂N₃O₄S | 437.468 g/mol |
| 1-{[2-(1,1-Difluoroethyl)-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]sulfonyl}-N-ethyl-1H-pyrrole-3-carboxamide | C₂₂H₂₆F₂N₄O₄S | 480.537 g/mol |
| 1-{[2-(1,1-dimethylpropyl)-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]sulfonyl}-N-isopropyl-1H-pyrrole-3-carboxamide | C₂₆H₃₆N₄O₄S | 500.665 g/mol |
| 1-{[2-(1,1-dimethylpropyl)-1-(tetrahydro-2H-pyran-4-ylmethyl)-1H-benzimidazol-5-yl]sulfonyl}-N-methyl-1H-pyrrole-3-carboxamide | C₂₄H₃₂N₄O₄S | 472.611 g/mol |
| 1-{[2-(4-Tert-butylthiazol-2-yl)benzofuran-5-yl]methyl}-5-(chloromethyl)indole-3-carbonitrile | C₂₆H₂₂ClN₃OS | 460.002 g/mol |
| 1-{[2-(4-Tert-butylthiazol-2-yl)benzofuran-5-yl]methyl}-5-(hydroxymethyl)indole-3-carbonitrile | C₂₆H₂₃N₃O₂S | 441.556 g/mol |