| 1-[(trifluoromethyl)sulphonyl]-1H-imidazole | C₄H₃F₃N₂O₂S | 200.141 g/mol |
| 1-[(Trifluoromethylsulfonyloxy)methyl]adamantane | C₁₂H₁₇F₃O₃S | 298.326 g/mol |
| 1-[(Z)-1-(4-chlorophenyl)prop-1-enyl]-1-(4-methoxyphenyl)-3-(6-methoxy-2-pyridinyl)-3-methylurea | C₂₄H₂₄ClN₃O₃ | 437.927 g/mol |
| 1-[(Z)-1-(4-chlorophenyl)prop-1-enyl]-1-(4-methoxyphenyl)-3-methylurea | C₁₈H₁₉ClN₂O₂ | 330.815 g/mol |
| 1-[({4-[(3-Chloro-2-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}methyl)(ethyl)amino]cyclopropanecarboxylic acid | C₂₂H₂₂ClFN₄O₃ | 444.894 g/mol |
| 1-[({4-[(3-Chloro-2-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}methyl)(methyl)amino]cyclopropanecarboxylic acid | C₂₁H₂₀ClFN₄O₃ | 430.867 g/mol |
| 1-[({4-[(3-Chloro-2-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}methyl)amino]cyclopropanecarboxylic acid | C₂₀H₁₈ClFN₄O₃ | 416.84 g/mol |
| 1-[({[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methyl}amino)carbonyl]cyclopropanecarboxylic acid | C₂₁H₂₉N₅O₄ | 415.494 g/mol |
| 1-[1'-benzyl-1-(5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)spiro[2H-indole-3,4'-piperidine]-4-yl]ethanol | C₂₉H₃₄N₄O | 454.618 g/mol |
| 1-[1,1-Dimethylethoxycarbonyl]-4-[3-(1-methylpropyl)amino-2-pyridinyl]piperazine | C₁₈H₃₀N₄O₂ | 334.464 g/mol |
| 1-[1,3,4]Oxadiazole-2-yl-3-phenylpropylamine | C₁₁H₁₃N₃O | 203.245 g/mol |
| 1-[1,5-Di-(bicyclo[2.2.2]oct-2-yl)-3-pentyl]-5-(2,3-dihydroxypropyl)-1,5,9-triazanonane | C₃₀H₅₇N₃O₂ | 491.805 g/mol |
| 1-[1,5-Di-(bicyclo[2.2.2]oct-2-yl)-3-pentyl]-5-(2,3-dihydroxypropyl)-9,9-di-(2,3-dihydroxypropyl)-1,5,9-triazanonane | C₃₆H₆₉N₃O₆ | 639.963 g/mol |
| 1-[1,8]Naphthyridin-4-ylethanone | C₁₀H₈N₂O | 172.187 g/mol |
| 1-[1-(1-Benzothien-3-yl)-4-piperidinyl]-4-(2-methoxyphenyl)piperazine | C₂₄H₂₉N₃OS | 407.583 g/mol |
| 1-[1-(1-benzyl-2-methyl-1H-indole-3-carbonyl)-piperidin-4-yl]-1,3-dihydro-benzoimidazol-2-one | C₂₉H₂₈N₄O₂ | 464.569 g/mol |
| 1-[1-(1-methoxycarbonylpiperidin-4-yl)-piperidin-4-yl]-3-acetyl-1,3-dihydro-2H-benzimidazol-2-one | C₂₁H₂₈N₄O₄ | 400.479 g/mol |
| 1-[1-(1-methoxycarbonylpiperidin-4-yl)piperidin-4-yl]-1,3-dihydro-2H-benzimidazol-2-one | C₁₉H₂₆N₄O₃ | 358.442 g/mol |
| 1-[1-(1-Methylpiperidin-4-yl)-1-phenylethyl]piperazine | C₁₈H₂₉N₃ | 287.451 g/mol |
| 1-[1-(1H-2-imidazolylmethyl)-4-piperidyl]-3-iodo-1H-pyrazolo[3,4-d]pyrimidin-4-amine | C₁₄H₁₇IN₈ | 424.25 g/mol |
| 1-[1-(2,4-Difluorophenethyl)-piperdin-4-yl]-6-bromoindoline | C₂₁H₂₃BrF₂N₂ | 421.329 g/mol |
| 1-[1-(2,4-Dimethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]ethan-1-one | C₁₆H₁₉NO₃ | 273.332 g/mol |
| 1-[1-(2,6-dioxo-1,3-dipropyl-7H-purin-8-yl)cyclopentyl]-3-propylurea | C₂₀H₃₂N₆O₃ | 404.515 g/mol |
| 1-[1-(2-[3-Indolyl]ethyl)piperid-4-yl]-3-cyclohexyl urea | C₂₂H₃₂N₄O | 368.525 g/mol |
| 1-[1-(2-chloro-phenyl)-5-(4-chloro-phenyl)-4-methyl-1H-pyrazole-3-carbonyl]-4-phenyl-piperidine-4-carboxylic acid ethyl ester | C₃₁H₂₉Cl₂N₃O₃ | 562.497 g/mol |
| 1-[1-(2-Chloro-phenyl)-cyclopropyl]-6-fluoro-2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-ol | C₁₉H₁₉ClFNO | 331.818 g/mol |
| 1-[1-(2-Chloro-phenyl)-ethyl]-7-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-1,2,3,4-tetrahydro-thieno[3,2-e][1,4]diazepin-5-one | C₂₁H₂₆BClN₂O₃S | 432.782 g/mol |
| 1-[1-(2-Chloro-phenyl)-ethyl]-7-imidazo[1,2-a]pyridin-3-yl-1,2,3,4-tetrahydro-thieno[3,2-e][1,4]diazepin-5-one | C₂₂H₁₉ClN₄OS | 422.941 g/mol |
| 1-[1-(2-Chloro-phenyl)cyclobutyl]-7-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinoline | C₂₁H₂₄ClNO | 341.882 g/mol |
| 1-[1-(2-chlorophenyl)-3,3-dimethylcyclobutyl]-6-methoxy-2-methyl-3,4-dihydro-1H-isoquinolin-7-ol | C₂₃H₂₈ClNO₂ | 385.935 g/mol |
| 1-[1-(2-Chlorophenyl)cyclobutyl]-7-methoxy-1,2,3,4-tetrahydroisoquinoline | C₂₀H₂₂ClNO | 327.855 g/mol |
| 1-[1-(2-Chlorophenyl)cyclopropyl]-6-fluoro-7-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinoline | C₂₀H₂₁ClFNO | 345.845 g/mol |
| 1-[1-(2-Chlorophenyl)cyclopropyl]-7-methoxy-3,4-dihydroisoquinoline | C₁₉H₁₈ClNO | 311.812 g/mol |
| 1-[1-(2-Cyanophenyl)cyclobutyl]-6,7-dimethoxy-3,4-dihydroisoquinoline | C₂₂H₂₂N₂O₂ | 346.43 g/mol |
| 1-[1-(2-Cyclopropylacetyl)pyrrolidin-3-yl]-3-[2-fluoro-4-[4-[[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]methyl]piperazine-1-carbonyl]phenyl]urea | C₃₁H₃₄F₇N₅O₄ | 673.63 g/mol |
| 1-[1-(2-fluoroethyl)-1H-pyrazol-4-yl]-2-[3-(2-fluoropyridin-3-yl)phenyl]ethane-1,2-dione | C₁₈H₁₃F₂N₃O₂ | 341.317 g/mol |
| 1-[1-(2-Hydroxyethyl)indazol-5-yl]-4-phenylmethoxypyridin-2-one | C₂₁H₁₉N₃O₃ | 361.401 g/mol |
| 1-[1-(2-Imidazol-1-yl-6-methyl-pyrimidin-4-yl)-ethyl]-pyrrolidine-2-carboxylic acid (benzo[1,3]dioxol-5-ylmethyl)-amide | C₂₃H₂₆N₆O₃ | 434.5 g/mol |
| 1-[1-(2-Methylindol-3-ylethyl)piperazin-4-yl]-3-(3,5-dimethoxyphenyl)urea | C₂₄H₃₁N₅O₃ | 437.544 g/mol |
| 1-[1-(2-Methylsulfanylphenyl)-4-phenylmethoxypentan-3-yl]imidazole-4-carboxamide | C₂₃H₂₇N₃O₂S | 409.555 g/mol |
| 1-[1-(2-Oxo-1,3-benzothiazol-3-yl)-4-phenylmethoxypentan-3-yl]imidazole-4-carboxamide | C₂₃H₂₄N₄O₃S | 436.537 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-5-(2,2-dimethylbutanoyl)-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-ethoxycarbonylphenyl)urea | C₃₅H₄₀N₄O₆ | 612.727 g/mol |
| 1-[1-(2-Toluoylmethyl)-2-oxo-5-(2-methylpentanoyl)-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-ethoxycarbonylphenyl)urea | C₃₅H₄₀N₄O₆ | 612.727 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-5-(2-thenoyl)-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-ethoxycarbonylphenyl)urea | C₃₄H₃₂N₄O₆S | 624.719 g/mol |
| 1-[1-(2-Toluoylmethyl)-2-oxo-5-benzyloxycarbonyl-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-ethoxycarbonylphenyl)urea | C₃₇H₃₆N₄O₇ | 648.716 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-5-cyclohexyl-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-ethoxycarbonylphenyl)urea | C₃₅H₄₀N₄O₅ | 596.728 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-5-cyclohexylcarbonyl-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-ethoxycarbonylphenyl)urea | C₃₆H₄₀N₄O₆ | 624.738 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-5-phenyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-methylphenyl)urea | C₃₂H₃₀N₄O₃ | 518.617 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-5-pivaloyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-benzyloxycarbonylphenyl)urea | C₃₈H₃₈N₄O₆ | 646.744 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-5-pivaloyl-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-methoxycarbonyl-4-fluorophenyl)urea | C₃₃H₃₅FN₄O₆ | 602.663 g/mol |
| 1-[1-(2-toluoylmethyl)-2-oxo-8-methyl-1,3,4,5-tetrahydro-2H-1,5-benzodiazepin-3-yl]-3-(3-ethoxycarbonylphenyl)urea | C₂₉H₃₀N₄O₅ | 514.582 g/mol |
| 1-[1-(2-trimethylsilanyl-ethoxymethyl)-1H-imidazol-4-yl]-cyclopropylamine | C₁₂H₂₃N₃OSi | 253.422 g/mol |
| 1-[1-(3,3-Dimethyl-2-oxopentyl)-6-methoxy-1H-indazol-3-yl]-2-methylprop-1-en-1-yl dimethyl phosphate | C₂₁H₃₁N₂O₆P | 438.461 g/mol |
| 1-[1-(3,4-dichloro-phenyl)-1H-imidazol-4-ylmethyl]-1H-imidazole-2-carbaldehyde | C₁₄H₁₀Cl₂N₄O | 321.167 g/mol |
| 1-[1-(3,4-Dichlorophenyl)cyclobutyl]ethylamine | C₁₂H₁₅Cl₂N | 244.165 g/mol |
| 1-[1-(3,4-Difluorophenethyl)-piperidin-4-yl]indoline | C₂₁H₂₄F₂N₂ | 342.433 g/mol |
| 1-[1-(3,4-Dihydro-2H-1,5-benzodioxepin-7-ylsulfonyl)-5-methoxy-1H-indol-4-yl]-N,N-dimethylmethanamine | C₂₁H₂₄N₂O₅S | 416.499 g/mol |
| 1-[1-(3,4-Dimethoxyphenylsulfanyl)-5-phenylpentyl]-cyclopentanecarboxylic acid | C₂₅H₃₂O₄S | 428.594 g/mol |
| 1-[1-(3,4-Dimethoxyphenylsulfanyl)-5-phenylpentyl]cyclopentane carboxylic acid hydroxyamide | C₂₅H₃₃NO₄S | 443.609 g/mol |
| 1-[1-(3,5-dichloro-benzyl)-1H-imidazol-2-yl]-2-(3-methoxy-phenyl)-ethanol | C₁₉H₁₈Cl₂N₂O₂ | 377.271 g/mol |
| 1-[1-(3,5-Dichloro-benzyl)-1H-imidazol-2-yl]-2-(3-methoxy-phenyl)-ethanone | C₁₉H₁₆Cl₂N₂O₂ | 375.255 g/mol |
| 1-[1-(3-Aminophenyl)-3-tert-butylpyrazol-5-yl]-3-(4-pyridin-4-ylsulfanylphenyl)urea | C₂₅H₂₆N₆OS | 458.591 g/mol |
| 1-[1-(3-Bromophenoxy)-4-hydroxypentan-3-yl]imidazole-4-carboxamide | C₁₅H₁₈BrN₃O₃ | 368.231 g/mol |
| 1-[1-(3-Cyclopentyloxy-4-methoxy-phenyl)-cyclopropylmethyl]-1,3-dihydro-imidazol-2-one | C₁₉H₂₄N₂O₃ | 328.412 g/mol |
| 1-[1-(3-Fluorophenethyl)piperdin-4-yl]-6-acetamidomethylindoline | C₂₄H₃₀FN₃O | 395.522 g/mol |
| 1-[1-(3-Methoxy-4-nitro-phenyl)-piperidin-4-ylmethyl]-4-methyl-piperazine | C₁₈H₂₈N₄O₃ | 348.447 g/mol |
| 1-[1-(3-tert-Butoxy-2-pyrazinylmethyl)-4-methylpiperidin-4-yl]-2-(2-fluorophenyl)ethanone | C₂₃H₃₀FN₃O₂ | 399.51 g/mol |
| 1-[1-(3-tert-Butoxy-2-pyrazinylmethyl)piperidin-4-yl]-2-(2-fluorophenyl)ethanone | C₂₂H₂₈FN₃O₂ | 385.483 g/mol |
| 1-[1-(3-Tert-butoxy-2-pyrazinylmethyl)piperidin-4-yl]-2-(2-methoxyphenyl)ethanone | C₂₃H₃₁N₃O₃ | 397.519 g/mol |
| 1-[1-(4,5-Diphenyloxazol-2-yl)ethylamino]-1,2,3,4-tetrahydro-5-ethoxycarbonylmethoxynaphthalene | C₃₁H₃₂N₂O₄ | 496.607 g/mol |
| 1-[1-(4-Acetamidomethylphenethyl)piperidin-4-yl]indoline | C₂₄H₃₁N₃O | 377.532 g/mol |
| 1-[1-(4-Amino-6,7-dimethoxyquinazolin-2-yl)piperidin-4-yl]-4,4-dimethylpiperidine-2,6-dione | C₂₂H₂₉N₅O₄ | 427.505 g/mol |
| 1-[1-(4-Amino-benzyl)-pyrrolidin-2-yl]-ethanol | C₁₃H₂₀N₂O | 220.316 g/mol |
| 1-[1-(4-Aminocyclohexanecarbonyl)-4-(4-fluorophenyl)pyrrolidin-3-yl]-3-[3,5-bis(trifluoromethyl)phenyl]-1,3-dimethylurea | C₂₈H₃₁F₇N₄O₂ | 588.568 g/mol |
| 1-[1-(4-Aminomethylphenethyl)piperidin-4-yl]indoline | C₂₂H₂₉N₃ | 335.495 g/mol |
| 1-[1-(4-Aminopiperidin-1-yl)propan-2-yl]piperidin-4-ol | C₁₃H₂₇N₃O | 241.379 g/mol |
| 1-[1-(4-Bromo-2,6-dimethylphenyl)-3,5-diethyl-1H-pyrazol-4-ylmethyl]-naphthalene-2-ol | C₂₆H₂₇BrN₂O | 463.419 g/mol |
| 1-[1-(4-Bromophenyl)ethyl]-4-phenylpiperidin-2-one | C₁₉H₂₀BrNO | 358.279 g/mol |
| 1-[1-(4-Bromophenyl)ethyl]piperazine | C₁₂H₁₇BrN₂ | 269.186 g/mol |
| 1-[1-(4-Cyano-benzyl)-2-oxocyclohexyl]-3-(3,5-dichlorophenyl)-urea | C₂₁H₁₉Cl₂N₃O₂ | 416.308 g/mol |
| 1-[1-(4-Cyanophenethyl)piperidin-4-yl]indoline | C₂₂H₂₅N₃ | 331.463 g/mol |
| 1-[1-(4-cyanophenyl)-3-(4-fluorophenyl)-2-hydroxypropyl]-1H-imidazole | C₁₉H₁₆FN₃O | 321.355 g/mol |
| 1-[1-(4-Cyanophenyl)-4-(4-fluorophenyl)butyl]-1,2,4-triazole | C₁₉H₁₇FN₄ | 320.371 g/mol |
| 1-[1-(4-Ethoxyphenyl)-2,5-dimethyl-1H-pyrrol-3-yl]ethan-1-one | C₁₆H₁₉NO₂ | 257.333 g/mol |
| 1-[1-(4-ethoxyphenyl)-5-fluorobenzimidazol-2-yl]-N-(thian-4-ylmethyl)ethanamine | C₂₃H₂₈FN₃OS | 413.562 g/mol |
| 1-[1-(4-Ethoxyphenyl)-5-fluorobenzimidazol-2-yl]ethanamine | C₁₇H₁₈FN₃O | 299.349 g/mol |
| 1-[1-(4-Fluoro-benzyl)-piperidin-4-yl]-4-(4-methanesulfonyl-phenoxy)-1H-pyrazolo[3,4-d]-pyrimidine | C₂₄H₂₄FN₅O₃S | 481.553 g/mol |
| 1-[1-(4-Fluorophenethyl)piperdin-4-yl]-5-chloro-6-aminoindoline | C₂₁H₂₅ClFN₃ | 373.903 g/mol |
| 1-[1-(4-Fluorophenethyl)piperidin-4-yl]-6-aminoindoline | C₂₁H₂₆FN₃ | 339.458 g/mol |
| 1-[1-(4-Fluorophenethyl)piperidin-4-yl]-6-aminomethylindole | C₂₂H₂₆FN₃ | 351.469 g/mol |
| 1-[1-(4-Fluorophenethyl)piperidin-4-yl]-6-aminomethylindoline | C₂₂H₂₈FN₃ | 353.485 g/mol |
| 1-[1-(4-Fluorophenethyl)piperidin-4-yl]-6-bromoacetamidomethylindole | C₂₄H₂₇BrFN₃O | 472.402 g/mol |
| 1-[1-(4-Fluorophenethyl)piperidin-4-yl]-6-chloromethylindoline | C₂₂H₂₆ClFN₂ | 372.915 g/mol |
| 1-[1-(4-Fluorophenethyl)piperidin-4-yl]-6-cyanoindoline | C₂₂H₂₄FN₃ | 349.453 g/mol |
| 1-[1-(4-Fluorophenethyl)piperidin-4-yl]-6-hydroxyiminomethylindoline | C₂₂H₂₆FN₃O | 367.468 g/mol |
| 1-[1-(4-Fluorophenyl)-2-hydroxyethyl]-3-[[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]methylidene]piperidin-2-one | C₂₅H₂₆FN₃O₃ | 435.499 g/mol |
| 1-[1-(4-Fluorophenyl)indazol-5-yl]-2-methyl-1-(1-prop-2-enylindol-3-yl)propan-1-ol | C₂₈H₂₆FN₃O | 439.534 g/mol |
| 1-[1-(4-Fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-amine | C₂₃H₂₂FN₃O₂ | 391.446 g/mol |
| 1-[1-(4-Fluorophenyl)indazol-5-yl]oxy-1-phenylpropan-2-amine | C₂₂H₂₀FN₃O | 361.42 g/mol |
| 1-[1-(4-fluorophenylmethyl)-1H-benzimidazol-2-yl]-1,5-diazacyclooctane | C₂₀H₂₃FN₄ | 338.43 g/mol |