| 1-[5-Methyl-2-(2-methyl-4-pyridinyl)pyrazol-3-yl]-4-[2-(trifluoromethyl)phenyl]sulfonylpyrrolidine-2-carboxylic acid | C₂₂H₂₁F₃N₄O₄S | 494.495 g/mol |
| 1-[5-methyl-2-(3-pyridinyl)-1H-imidazol-4-yl]ethanone | C₁₁H₁₁N₃O | 201.229 g/mol |
| 1-[5-methylaminomethyl-1-(3-methyl-butyl)-1H-benzoimidazol-2-ylmethyl]-3-isopropyl-1,3-dihydro-benzoimidazol-2-one | C₂₅H₃₃N₅O | 419.573 g/mol |
| 1-[5-t-butyl-2-(3-chloromethyl-phenyl)-2H-pyrazol-3-yl]-3-(4-fluoro-phenyl)-urea | C₂₁H₂₂ClFN₄O | 400.885 g/mol |
| 1-[5-tert-Butyl-2-(2-hydroxy-ethyl)-2H-pyrazol-3-yl]-3-{4-[7-(4-methanesulfonyl-phenyl)-imidazo[1,2-a]pyridin-3-yl]-benzyl}-urea | C₃₁H₃₄N₆O₄S | 586.718 g/mol |
| 1-[6,6-Dioxido-2-(2,4,5-trifluorophenyl)-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one | C₁₇H₁₅F₃N₄O₃S | 412.393 g/mol |
| 1-[6,7-Dimethyl-5-(tetrahydro-pyran-2-yloxy)-benzofuran-2-yl]-ethanone | C₁₇H₂₀O₄ | 288.343 g/mol |
| 1-[6-(1,1,1,2,3,3,3-Heptafluoropropan-2-yl)-3-(pyridin-3-ylmethylamino)-2,4-dihydroquinazolin-1-yl]ethanone | C₁₉H₁₇F₇N₄O | 450.358 g/mol |
| 1-[6-(1-Phenylethylamino)pyrazin-2-yl]benzimidazol-5-amine | C₁₉H₁₈N₆ | 330.395 g/mol |
| 1-[6-(2,4-Difluoro-phenoxy)-3-iodo-1H-pyrazolo[3,4-d]pyrimidin-4-ylamino]-propan-2-ol | C₁₄H₁₂F₂IN₅O₂ | 447.183 g/mol |
| 1-[6-(2,5-Dimethylpyrrol-1-yl)pyridin-3-yl]-2-propylaminoethanol | C₁₆H₂₃N₃O | 273.38 g/mol |
| 1-[6-(2-Chloro-4-methoxy-5-methyl-phenyl)-5-methyl-pyrazin-2-yl]-1H-benzotriazole | C₁₉H₁₆ClN₅O | 365.824 g/mol |
| 1-[6-(2-Chloro-4-methoxyphenoxy)hexyl]-3-methylimidazol-3-ium | C₁₇H₂₄ClN₂O₂+ | 323.844 g/mol |
| 1-[6-(2-Chloro-4-methyxyphenoxy)-hexyl]-imidazole | C₁₆H₂₁ClN₂O₂ | 308.809 g/mol |
| 1-[6-(2-Methylpropyl)-1,3-benzoxazol-2-yl]piperidine-2-carboxylic acid | C₁₇H₂₂N₂O₃ | 302.374 g/mol |
| 1-[6-(3,3-Dimethyl-but-1-enyl)-pyridin-3-ylmethyl]-3-hydroxy-1H-thieno[3,2-d]pyrimidine-2,4-dione | C₁₈H₁₉N₃O₃S | 357.435 g/mol |
| 1-[6-(3,5-dimethylpiperazin-1-yl)-5-methoxy-3,3-dimethyl-2H-indol-1-yl]ethanone | C₁₉H₂₉N₃O₂ | 331.46 g/mol |
| 1-[6-(3-Chloro-phenylamino)-pyrimidin-4-yl]-3-(2,5-dimethoxy-phenyl)-urea | C₁₉H₁₈ClN₅O₃ | 399.838 g/mol |
| 1-[6-(3-Dimethylamino-pyrrolidin-1-yl)-2-methyl-4-phenyl-quinolin-3-yl]-2,2,2-trifluoro-ethanone | C₂₄H₂₄F₃N₃O | 427.47 g/mol |
| 1-[6-(3-Methoxyphenyl)-5,8,10-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraen-5-yl]ethanone | C₁₉H₁₉N₃O₂ | 321.38 g/mol |
| 1-[6-(3-trifluoromethyl-1-trityl-1H-pyrazol-4-yl)quinolin-4-yl]-piperidine-4-carboxylic acid (4-fluorophenyl)methylamide | C₄₅H₃₇F₄N₅O | 739.817 g/mol |
| 1-[6-(4-Amino-2-fluorophenoxy)pyrimidin-4-yl]-3-(1-methylpiperidin-4-yl)urea | C₁₇H₂₁FN₆O₂ | 360.393 g/mol |
| 1-[6-(4-Benzotriazol-2-yl-but-1-ynyl)-pyridin-2-yl]-ethanol | C₁₇H₁₆N₄O | 292.342 g/mol |
| 1-[6-(4-Benzotriazol-2-yl-but-1-ynyl)-pyridin-2-yl]-ethanone | C₁₇H₁₄N₄O | 290.326 g/mol |
| 1-[6-(4-Bromo-2-chloro-phenylamino)-7-fluoro-3-methyl-3H-benzoimidazol-5-yl]-2-hydroxy-ethanone | C₁₆H₁₂BrClFN₃O₂ | 412.646 g/mol |
| 1-[6-(4-Bromo-2-chloro-phenylamino)-7-fluoro-3-methyl-3H-benzoimidazol-5-yl]-2-methoxymethoxy-ethanol | C₁₈H₁₈BrClFN₃O₃ | 458.715 g/mol |
| 1-[6-(4-Bromo-2-chloro-phenylamino)-7-fluoro-3-methyl-3H-benzoimidazol-5-yl]-2-methoxymethoxy-ethanone | C₁₈H₁₆BrClFN₃O₃ | 456.699 g/mol |
| 1-[6-(4-Bromo-2-chloro-phenylamino)-7-fluoro-3H-benzoimidazol-5-yl]-2-ethoxy-ethanone | C₁₇H₁₄BrClFN₃O₂ | 426.673 g/mol |
| 1-[6-(4-Bromo-2-chloro-phenylamino)-7-fluoro-3H-benzoimidazol-5-yl]-2-methoxymethoxy-ethanol | C₁₇H₁₆BrClFN₃O₃ | 444.688 g/mol |
| 1-[6-(4-Bromo-2-chloro-phenylamino)-7-fluoro-3H-benzoimidazol-5-yl]-2-methoxymethoxy-ethanone | C₁₇H₁₄BrClFN₃O₃ | 442.672 g/mol |
| 1-[6-(4-Bromo-phenoxy)-pyridin-3-yl]-pyrrolidine-2,2-dicarboxylic acid diethyl ester | C₂₁H₂₃BrN₂O₅ | 463.328 g/mol |
| 1-[6-(4-Chloro-phenoxy)-pyridin-2-yl]-piperazine | C₁₅H₁₆ClN₃O | 289.766 g/mol |
| 1-[6-(4-Fluorophenyl)imidazo[2,1-b][1,3]oxazol-5-yl]ethanone | C₁₃H₉FN₂O₂ | 244.225 g/mol |
| 1-[6-(4-Hydroxy-3,5-dimethyl-phenyl)-3-methoxy-pyridazin-4-yl]-propan-1-one | C₁₆H₁₈N₂O₃ | 286.331 g/mol |
| 1-[6-(4-Imidazol-1-yl-phenoxy)-5-nitro-pyrimidin-4-yl]-piperidine-4-carboxylic acid ethyl ester | C₂₁H₂₂N₆O₅ | 438.444 g/mol |
| 1-[6-(4-Methanesulfonyl-phenylamino)-2-phenyl-pyrimidin-4-yl]-piperidin-4-ol | C₂₂H₂₄N₄O₃S | 424.526 g/mol |
| 1-[6-(4-Methoxyphenoxy)hexyl]-3-methyl-7-propylxanthine | C₂₂H₃₀N₄O₄ | 414.506 g/mol |
| 1-[6-(4-Phenyl-2-quinolyloxy)hexanoyl]pyrrolidine | C₂₅H₂₈N₂O₂ | 388.511 g/mol |
| 1-[6-(4-Vinyl-phenoxy)-pyridin-3-yl]-pyrrolidine-2,2-dicarboxylic acid diethyl ester | C₂₃H₂₆N₂O₅ | 410.47 g/mol |
| 1-[6-(5-Methyl-2-phenyl-4-oxazolylmethoxy)-3-pyridylmethyl]-4-phenyl-3-pyrrolecarbaldehyde | C₂₈H₂₃N₃O₃ | 449.51 g/mol |
| 1-[6-(5-{1-[4-(cyclopropylsulfonyl)phenyl]-2-(tetrahydro-2H-pyran-4-yl)ethyl}-1H-pyrrol-2-yl)pyridin-3-yl]ethanol | C₂₇H₃₂N₂O₄S | 480.63 g/mol |
| 1-[6-(6-Chloro-pyrazolo[1,5-a]pyrimidine-2-carbonyl)-7-methyl-4,5,6,7-tetrahydropyrrolo[2,3-c]pyridin-1-yl]-ethanone | C₁₇H₁₆ClN₅O₂ | 357.801 g/mol |
| 1-[6-(Azetidin-1-yl-methyl)-1,2,3,4-tetrahydro-isoquinolin-2-yl]-2,2,2-trifluoro-ethanone | C₁₅H₁₇F₃N₂O | 298.308 g/mol |
| 1-[6-(Cyclopropylmethoxy)-3-phenanthryl]-2-methylpropan-2-ol | C₂₂H₂₄O₂ | 320.432 g/mol |
| 1-[6-(N-tert-Butoxycarbonylamino)-1-hexyl]-1,2-dihydroquinoline-2-one | C₂₀H₂₈N₂O₃ | 344.455 g/mol |
| 1-[6-(N-tert-Butoxycarbonylamino)-1-hexyl]-imidazole | C₁₄H₂₅N₃O₂ | 267.373 g/mol |
| 1-[6-(Nonyloxy)-2,3-dihydro-1H-inden-1-YL]piperazine | C₂₂H₃₆N₂O | 344.543 g/mol |
| 1-[6-(Trifluoromethyl)pyridin-2-yl]piperazine | C₁₀H₁₂F₃N₃ | 231.221 g/mol |
| 1-[6-(Trifluoromethyl)pyridin-3-yl]ethan-1-one | C₈H₆F₃NO | 189.136 g/mol |
| 1-[6-(Tritylamino)hexyl]pyrimidine-2,4-dione | C₂₉H₃₁N₃O₂ | 453.586 g/mol |
| 1-[6-({4-[2-Hydroxypropyl]phenyl}amino)-5-nitro-3-pyridinyl]ethanone | C₁₆H₁₇N₃O₄ | 315.329 g/mol |
| 1-[6-[3-(Dimethylamino)anilino]pyrimidin-4-yl]-1-methyl-3-(2-methyl-5-nitrophenyl)urea | C₂₁H₂₃N₇O₃ | 421.461 g/mol |
| 1-[6-Amino-5-chloro-2-(methoxy)-3-pyridinyl]-3-(1-butyl-4-piperidinyl)-1-propanone | C₁₈H₂₈ClN₃O₂ | 353.894 g/mol |
| 1-[6-Azepan-1-yl-4-(4-fluoro-phenyl)-2-methyl-quinolin-3-yl]-2,2,2-trifluoro-ethanone | C₂₄H₂₂F₄N₂O | 430.445 g/mol |
| 1-[6-benzyl-5-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)-2-pyridinyl]-4-methoxypyrrolidin-3-ol | C₂₃H₂₉N₃O₂ | 379.504 g/mol |
| 1-[6-Benzyl-5-[2-(1-piperidin-1-ylcyclohexyl)ethynyl]-2-pyridinyl]-4-methoxypyrrolidin-3-ol | C₃₀H₃₉N₃O₂ | 473.661 g/mol |
| 1-[6-Benzyloxy-2-hydroxy-3-(5-methyl-7-nitroindan-4-yloxy)phenyl]ethanone | C₂₅H₂₃NO₆ | 433.46 g/mol |
| 1-[6-Benzyloxy-2-methoxy-3-(5-methyl-7-nitroindan-4-yloxy)phenyl]ethanone | C₂₆H₂₅NO₆ | 447.487 g/mol |
| 1-[6-Bromo-4-(4-fluoro-phenyl)-2-methyl-quinolin-3-yl]-2,2,2-trifluoro-ethanone | C₁₈H₁₀BrF₄NO | 412.18 g/mol |
| 1-[6-Bromo-4-(4-methanesulfonyl-phenyl)-2-methyl-quinolin-3-yl]-2,2,2-trifluoro-ethanone | C₁₉H₁₃BrF₃NO₃S | 472.282 g/mol |
| 1-[6-Chloro-1-(3,5-difluoro-benzyl)-1H-indol-3-yl]-2,2,2-trifluoro-ethanone | C₁₇H₉ClF₅NO | 373.708 g/mol |
| 1-[6-Chloro-1-(3,5-difluoro-phenyl)-1H-indol-3-yl]-2,2,2-trifluoro-ethanone | C₁₆H₇ClF₅NO | 359.681 g/mol |
| 1-[6-chloro-1-(3-methyl-butyl)-1H-indol-3-yl]-2,2,2-trifluoro-ethanone | C₁₅H₁₅ClF₃NO | 317.738 g/mol |
| 1-[6-Chloro-2-[1-(4-fluorophenyl)ethylamino]pyrimidin-4-yl]-4-(hydroxymethyl)piperidin-4-ol | C₁₈H₂₂ClFN₄O₂ | 380.851 g/mol |
| 1-[6-Chloro-2-[1-(4-fluorophenyl)ethylamino]pyrimidin-4-yl]pyrrolidin-3-ol | C₁₆H₁₈ClFN₄O | 336.798 g/mol |
| 1-[6-cyano-7-(4-cyanophenyl)-5-methyl-4-[3-(trifluoromethyl)phenyl]-7H-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-3-ethylurea | C₂₄H₁₉F₃N₈O | 492.465 g/mol |
| 1-[6-Fluoro-2-(4-chlorophenyl)-4-quinolinyl]-N-methyl-4-piperidinecarboxamide | C₂₂H₂₁ClFN₃O | 397.881 g/mol |
| 1-[6-Hydrazinyl-4-(methylamino)pyridazin-3-yl]propan-2-ol | C₈H₁₅N₅O | 197.242 g/mol |
| 1-[6-methoxy-4-[(3-methyl-1H-indol-5-yl)oxy]quinazolin-7-yl]oxy-3-(3-pyrrolidin-1-ylpropylamino)propan-2-ol | C₂₈H₃₅N₅O₄ | 505.619 g/mol |
| 1-[6-Methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-yl]-3-(1-phenylethyl)urea | C₂₅H₃₁N₅O₃ | 449.555 g/mol |
| 1-[6-Methoxy-pyridin-3-ylmethoxy]-naphthalene-2-carboxylic acid | C₁₈H₁₅NO₄ | 309.321 g/mol |
| 1-[6-Methoxypyridin-3-yl]-1-[1-(pyridin-3-yl)indazol-5-yl]oxypropan-2-amine | C₂₁H₂₁N₅O₂ | 375.432 g/mol |
| 1-[6-Methyl-2-phenyl-4-quinolinyl]-4-piperidinecarboxamide | C₂₂H₂₃N₃O | 345.446 g/mol |
| 1-[6-Methyl-5-(trifluoromethyl)pyridin-2-yl]azetidin-3-amine | C₁₀H₁₂F₃N₃ | 231.221 g/mol |
| 1-[7,8-Dimethoxy-1,3,4,5-tetrahydro-2H-3-benzazepin-1,2-dion-3-yl]-3-[N-methyl-N-(6,7-dimethoxy-1,2,3,4-tetrahydronaphth-2-yl)-amino]-propane | C₂₈H₃₆N₂O₆ | 496.604 g/mol |
| 1-[7,8-Dimethoxy-1,3,4,5-tetrahydro-2H-3-benzazepin-2-on-3-yl]-3-[N-(6,7-dimethoxy-1,2,3,4-tetrahydronaphth-2-yl)-amino]-propane | C₂₇H₃₆N₂O₅ | 468.594 g/mol |
| 1-[7,8-Dimethoxy-1,3,4,5-tetrahydro-2H-3-benzazepin-2-on-3-yl]-3-[N-benzyl-N-(6,7-dimethoxy-1,2,3,4-tetrahydronaphth-2-yl)-amino]-propane | C₃₄H₄₂N₂O₅ | 558.719 g/mol |
| 1-[7,8-Dimethoxy-1,3,4,5-tetrahydro-2H-3-benzazepin-2-on-3-yl]-3-[N-methyl-N-(2-{4-amino-3,5-dichloro-phenyl}-ethyl)-amino]-propane | C₂₄H₃₁Cl₂N₃O₃ | 480.436 g/mol |
| 1-[7,8-Dimethoxy-1,3,4,5-tetrahydro-2H-3-benzazepin-2-on-3-yl]-3-[N-methyl-N-(5-methoxy-1,2,3,4-tetrahydronaphth-2-yl)-amino]-propane | C₂₇H₃₆N₂O₄ | 452.595 g/mol |
| 1-[7,8-dimethoxy-1,3-dihydro-2H-3-benzazepin-2-on-3-yl]-3-[N-methyl-N-(2-{4-amino-3,5-dichloro-phenyl}-ethyl)-amino]-propane | C₂₄H₂₉Cl₂N₃O₃ | 478.42 g/mol |
| 1-[7-(1,5-dimethyl-1H-[1,2,4]triazol-3-yl)-imidazo[1,2-a]pyridin-2-yl]-3-ethyl-urea | C₁₄H₁₇N₇O | 299.338 g/mol |
| 1-[7-(3-Chloro-phenylamino)-1,3-dimethyl-1H-pyrrolo[2,3-c]pyridin-4-yl]-1-morpholin-4-yl-methanone | C₂₀H₂₁ClN₄O₂ | 384.867 g/mol |
| 1-[7-(4-Fluorophenyl)-17,20-dihydroxy-2,18-dimethyl-6,7-diazapentacyclo[11.7.0.02,10.04,8.014,18]icosa-4(8),5,9-trien-17-yl]-2-hydroxyethanone | C₂₈H₃₃FN₂O₄ | 480.58 g/mol |
| 1-[7-(4-Hydroxyphenyl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl]-3-(6-methylheptan-2-yl)urea | C₂₀H₂₆N₆O₂ | 382.468 g/mol |
| 1-[7-(5-Cyano-pyridin-2-yl)-5-pyridin-3-yl-benzothiazol-2-yl]-3-ethyl-urea | C₂₁H₁₆N₆OS | 400.467 g/mol |
| 1-[7-(6-Chloro-indole-1-sulfonyl)-4,4-dimethyl-3,4-dihydro-1H-isoquinolin-2-yl]-ethanone | C₂₁H₂₁ClN₂O₃S | 416.93 g/mol |
| 1-[7-(Bis{[2-(trimethylsilyl)ethoxy]methyl}amino)pyrazolo[1,5-a]pyrimidin-5-yl]ethanone | C₂₀H₃₆N₄O₃Si₂ | 436.705 g/mol |
| 1-[7-(Chloro)-2-(4-methoxyphenyl)pyrazolo[1,5-a]pyridin-3-yl]ethanone | C₁₆H₁₃ClN₂O₂ | 300.745 g/mol |
| 1-[7-(Cyclopentylamino)-2-(4-fluorophenyl)pyrazolo[1,5-a]pyridin-3-yl]ethanone | C₂₀H₂₀FN₃O | 337.398 g/mol |
| 1-[7-[1-(2-dimethylaminoethyl)pyrazol-3-yl]-4-fluoro-1H-pyrrolo[2,3-c]pyridin-3-yl]-2-[4-(1-phenyltetrazol-5-yl)piperazin-1-yl]ethane-1,2-dione | C₂₇H₂₈FN₁₁O₂ | 557.594 g/mol |
| 1-[7-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3,4-dihydro-1H-isoquinolin-2-yl]-2-pyrrolidin-3-ylethanone | C₂₄H₃₃N₇O | 435.576 g/mol |
| 1-[7-[2-Hydroxy-3-[4-(2-methylphenyl)piperazin-1-yl]propoxy]-1-benzofuran-2-yl]ethanone | C₂₄H₂₈N₂O₄ | 408.498 g/mol |
| 1-[7-Benzyloxy-8-hydroxy-1,3,4,5-tetrahydro-2H-3-benzazepin-2-on-3-yl]-3-[N-methyl-N-(2-{3,4-dimethoxy-phenyl}-ethyl)-amino]-propane | C₃₁H₃₈N₂O₅ | 518.654 g/mol |
| 1-[7-bromo-2-(ethoxymethyl)-1H-imidazo[4,5-c][1,5]naphthyridin-1-yl]-2-methylpropan-2-ol | C₁₆H₁₉BrN₄O₂ | 379.258 g/mol |
| 1-[7-Bromo-5-fluoro-3-(3-fluoro-benzyl)-benzofuran-2-yl]-ethanone | C₁₇H₁₁BrF₂O₂ | 365.173 g/mol |
| 1-[7-Chloro-2-(2-furyl)pyrazolo[1,5-a]pyridin-3-yl]-2-propyn-1-ol | C₁₄H₉ClN₂O₂ | 272.691 g/mol |
| 1-[7-Chloro-2-(2-furyl)pyrazolo[1,5-a]pyridin-3-yl]-2-propyn-1-one | C₁₄H₇ClN₂O₂ | 270.675 g/mol |
| 1-[7-Chloro-3-(3,5-dimethyl-phenyl)-2-oxo-4-(2-piperidin-2-yl-ethoxy)-1,2-dihydro-quinolin-6-yl]-3-pyridin-4-yl-urea | C₃₀H₃₂ClN₅O₃ | 546.071 g/mol |
| 1-[7-chloro-4-(4-fluorophenyl)-2,2-dimethyl-2H-chromen-3-yl]ethanone | C₁₉H₁₆ClFO₂ | 330.786 g/mol |
| 1-[7-Chloro-6-[1-(3,5-difluoro-4-methoxyphenyl)ethylamino]-1,2,4,5-tetrahydro-3-benzazepin-3-yl]-2,2,2-trifluoroethanone | C₂₁H₂₀ClF₅N₂O₂ | 462.846 g/mol |