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Buchwald–Hartwig amination, record ord-5dfaf464504c42b7bafec75259e5a214

One recorded run of this reaction. Below is what the source recorded, and nothing added to it.

verified record11% yield recordedNot balanced as writtenFrom experimental reaction archive

Reactants and products as the record gives them. Reagents, catalysts and solvents are listed below rather than drawn.

Open this record in the Reaction LabThe atom map, the animation and the records that run the same transformation.

What was in the flask

RoleSpeciesFormulaYield
Reactant2,4-DichloropyridineC₅H₃Cl₂N
Reactant2-AminooxazoleC₃H₄N₂O
ReagentCesium carbonateCCs₂O₃
Catalyst1,1'-(9,9-Dimethyl-9H-xanthene-4,5-diyl)bis(1,1-diphenylphosphine)C₃₉H₃₂OP₂
CatalystPalladium (II) acetateC₄H₈O₄Pd
Solvent1,4-DioxaneC₄H₈O₂
ProductN-(4-chloro-2-pyridinyl)-1,3-oxazol-2-amineC₈H₆ClN₃O11.1%

The equation does not balance as written. That is usual for an experimental record: the source listed what it put in and what it measured, not a stoichiometric equation.

Conditions

Temperature
100 °C

Only the dimensions the source stated are listed. Anything absent here was not recorded, and it is not inferred from what the class usually needs.

Yield

  • 11% of N-(4-chloro-2-pyridinyl)-1,3-oxazol-2-amine.

Procedure

Copied from the source record, unedited

Palladium(II) acetate (11.38 mg, 0.05 mmol) was added in a single portion to a degassed solution of 9,9-dimethyl-4,5-bis(diphenylphosphino)xanthene (44.0 mg, 0.08 mmol), oxazol-2-amine (85 mg, 1.01 mmol), cesium carbonate (768 mg, 2.36 mmol),2,4-dichloropyridine (0.109 mL, 1.01 mmol), dioxane (4 mL) and DMSO (0.8 mL) and the resulting mixture was heated at 100 °C for 16 hours under a nitrogen atmosphere. Note: the reaction mixture was degassed by first combing the reagents (with the exception of Pd((OAc)2), sealing the vessel and carrying out three pump- purge cycles (vac-nitrogen). Dioxane was then added to this mixture via syringe, followed by the Pd(OAc)2 in a single portion and the vessel was heated for the required time as above. Solvent boiled dry from reaction overnight. Only DMSO

The source

This record comes from experimental reaction archive (ord-5dfaf464504c42b7bafec75259e5a214). Open the source and check it against what is on this page.

  • experimental reaction archive record ord-5dfaf464504c42b7bafec75259e5a214 from dataset "750 AstraZeneca ELN dataset" (url: https://chemrxiv.org/engage/chemrxiv/article-details/60c9e3f37792a23bfdb2d471). No atom mapping is provided by the source.

    experimental record · quality medium · source

experimental reaction record.

How to read this record

This is one experiment, not a rule. It says that on one occasion these species were combined under these conditions and this came out. It does not say the reaction will give the same result on your substrate, and nothing on the page has been generalised into a claim that it would.

The pathway is a separate question, kept on separate pages. A mechanism here is the canonical arrow pushing for a class, run on real structures and labelled rule-derived. It is not evidence, and this record is not a mechanism.