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Buchwald–Hartwig amination, record ord-cab6249a1023430399dca1061d293aa8

One recorded run of this reaction. Below is what the source recorded, and nothing added to it.

verified record3% yield recordedNot balanced as writtenFrom experimental reaction archive

Reactants and products as the record gives them. Reagents, catalysts and solvents are listed below rather than drawn.

Open this record in the Reaction LabThe atom map, the animation and the records that run the same transformation.

What was in the flask

RoleSpeciesFormulaYield
Reactant2,4-DichloropyridineC₅H₃Cl₂N
Reactant2-AminooxazoleC₃H₄N₂O
Reagentsodium phenoxideC₆H₅NaO
Catalyst1,1'-(9,9-Dimethyl-9H-xanthene-4,5-diyl)bis(1,1-diphenylphosphine)C₃₉H₃₂OP₂
CatalystBis(dibenzylideneacetone)palladiumC₅₁H₄₂O₃Pd₂
Solvent1,4-DioxaneC₄H₈O₂
ProductN-(4-chloro-2-pyridinyl)-1,3-oxazol-2-amineC₈H₆ClN₃O2.52%

The equation does not balance as written. That is usual for an experimental record: the source listed what it put in and what it measured, not a stoichiometric equation.

Conditions

Temperature
80 °C

Only the dimensions the source stated are listed. Anything absent here was not recorded, and it is not inferred from what the class usually needs.

Yield

  • 3% of N-(4-chloro-2-pyridinyl)-1,3-oxazol-2-amine.

Procedure

Copied from the source record, unedited

To a flask containing 2,4-dichloropyridine (0.109 mL, 1.01 mmol), sodium phenolate (177 mg, 1.52 mmol), TRIS(DIBENZYLIDENEACETONE)DIPALLADIUM(0) (11.60 mg, 0.01 mmol) and (9,9-dimethyl-9H-xanthene-4,5-diyl)bis(diphenylphosphine) (17.59 mg, 0.03 mmol) (Xantphos), was added degassed dioxane (4 mL) and the mixture allowed to stir under nitrogen atmosphere for 5 min. To this solution was added oxazol-2-amine (94 mg, 1.11 mmol) and the reaction mixture was heated to 80 °C for three hours. A 1H NMR was measured of the crude reaction after the solvent had been removed. **This indicated the presence of significant amounts of 2,4-dichloropyridine as well as 2-amino oxazole**. LCMS of the crude reaction mixture at t= 90 min and at t= 3 h showed the desired product was present. The crude reaction mi

The source

This record comes from experimental reaction archive (ord-cab6249a1023430399dca1061d293aa8). Open the source and check it against what is on this page.

  • experimental reaction archive record ord-cab6249a1023430399dca1061d293aa8 from dataset "750 AstraZeneca ELN dataset" (url: https://chemrxiv.org/engage/chemrxiv/article-details/60c9e3f37792a23bfdb2d471). No atom mapping is provided by the source.

    experimental record · quality medium · source

experimental reaction record.

How to read this record

This is one experiment, not a rule. It says that on one occasion these species were combined under these conditions and this came out. It does not say the reaction will give the same result on your substrate, and nothing on the page has been generalised into a claim that it would.

The pathway is a separate question, kept on separate pages. A mechanism here is the canonical arrow pushing for a class, run on real structures and labelled rule-derived. It is not evidence, and this record is not a mechanism.