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Buchwald–Hartwig amination, record ord-7a326b6af66842839478f845f091880c

One recorded run of this reaction. Below is what the source recorded, and nothing added to it.

verified record0% yield recordedNot balanced as writtenFrom experimental reaction archive

Reactants and products as the record gives them. Reagents, catalysts and solvents are listed below rather than drawn.

Open this record in the Reaction LabThe atom map, the animation and the records that run the same transformation.

What was in the flask

RoleSpeciesFormulaYield
Reactant3-Bromo-2,6-dichloropyridineC₅H₂BrCl₂N
ReactantMorpholineC₄H₉NO
Reagentsodium 2-methylpropan-2-olateC₄H₉NaO
Catalyst2-Dicyclohexylphosphino-2',6'-diisopropoxybiphenylC₃₀H₄₃O₂P
CatalystBis(dibenzylideneacetone)palladiumC₅₁H₄₂O₃Pd₂
SolventTetrahydrofuranC₄H₈O
Product4-(2,6-Dichloro-3-pyridinyl)morpholineC₉H₁₀Cl₂N₂O0%

The equation does not balance as written. That is usual for an experimental record: the source listed what it put in and what it measured, not a stoichiometric equation.

Conditions

Temperature
100 °C

Only the dimensions the source stated are listed. Anything absent here was not recorded, and it is not inferred from what the class usually needs.

Yield

  • 0% of 4-(2,6-Dichloro-3-pyridinyl)morpholine.

Procedure

Copied from the source record, unedited

sodium tert-butoxide (0.012 g, 0.13 mmol), were transfered to a microwave vial. Pd2dba3 (0.916 mg, 1.00 µmol), dicyclohexyl(2',6'-diisopropoxybiphenyl-2-yl)phosphine (0.933 mg, 2.00 µmol), (2-DICYCLOHEXYLPHOSPHINO-2',6'-DIISOPROPYL-1,1'-BIPHENYL)[2-(2-AMINOETHYL)PHENYL]PALLADIUM(II) (0.729 mg, 1.00 µmol) were added. 3-bromo-2,6-dichloropyridine (0.011 g, .05 mmol) in tetrahydrofuran (0.474 ml) was added. The vial was flushed with N2, sealed, and the reaction mix was heated on an oil bath at 100 °C. 2011-10-05 0900: interrupted, cooled- LC/MS, 5 min method, pH11: 1H NMR on crude:not good spectra. 2011-10-06 The mix was filtered thru Si-plug and conc. 1H NMR and COSY. Very complex. Lower rection temp and time needed. Discarded. \---- Info from -25: 2011-09-18 Lit. ref: ....B

The source

This record comes from experimental reaction archive (ord-7a326b6af66842839478f845f091880c). Open the source and check it against what is on this page.

  • experimental reaction archive record ord-7a326b6af66842839478f845f091880c from dataset "750 AstraZeneca ELN dataset" (url: https://chemrxiv.org/engage/chemrxiv/article-details/60c9e3f37792a23bfdb2d471). No atom mapping is provided by the source.

    experimental record · quality medium · source

experimental reaction record.

How to read this record

This is one experiment, not a rule. It says that on one occasion these species were combined under these conditions and this came out. It does not say the reaction will give the same result on your substrate, and nothing on the page has been generalised into a claim that it would.

The pathway is a separate question, kept on separate pages. A mechanism here is the canonical arrow pushing for a class, run on real structures and labelled rule-derived. It is not evidence, and this record is not a mechanism.